CEOs Publications

My research in the industry







PUBLICATIONS (Top 25 out of 50)

Asymmetric Synthesis of 1-Substituted 2-Azaspiro[3.3]heptanes: An Important  Motifs for Modern Drug Discovery.
Rajender Reddy Leleti* et. al.
Chem. Coumn. 2019, ASAP article.

Asymmetric Synthesis 1-Substituted 2,6-Diazaspiro[3.3]heptanes.
Rajender Reddy Leleti* et. al.
Organic Letters. 2019ASAP article.

Umpolung Synthesis of Vicinal Diamines: Diastereoselective Addi-tion of 2‑Azaallyl Anions to Davis–Ellman’s Imines.
Rajender Reddy Leleti* et. al.
Organic Letters.  2018, 20, 5423.

N-Arylation of carbamates through photosensitized nickel catalysis.
Rajender Reddy Leleti* et. al.
J. Org. Chem. 2018, 83, 13854.

Diastereoselective Addition of Anisoles to N-tert-Butanesulfinylimines via Four-Membered Lithiumcycles.
Rajender Reddy Leleti* et. al.
Chem. Coumn. 2018, 54, 7007

Asymmetric Synthesis of a-(diarylmethyl) alkyl amines through Regioselective Lithiation of a-Diarylmethanes and Diastereoselective Addition to Ellman’s Imines.
Rajender Reddy Leleti* et. al.
J. Org. Chem. 2018, 83, 6573

Chiral Bronsted Acid Catalysed Enantioselective Propargylation of Aldehydes with Allenyl  boronate.
Rajender Reddy Leleti*
Organic Letters 2012, 14, 1142.

Chiral Bronsted Acid Catalyzed Enantioselective Allenylation of Aldehydes.
Rajender Reddy Leleti*
Chem. Coumn. 2012, 48, 9189.

A Protocol for an Asymmetric Synthesis of γ-Amino Acids. 
Rajender Reddy Leleti* et. al.
J. Org. Chem.  2012, 77, 6296.

A Simple and Efficient Rhodium-Catalyzed Asymmetric Arylation of N-tert-Butanesulfinyl
Imines with Sodium Tetraarylborates.
Rajender Reddy Leleti* et. al.
J. Org. Chem2012, 77, 1095.

Asymmetric Synthesis of α-Amino Acids by Reduction of N-tert-Butanesulfinyl Ketimine Esters .
Rajender Reddy Leleti* et. al.
J. Org. Chem. 2011, 76, 3409.         

A Facile Asymmetric Synthesis of Either Enantiomer of 2-Substituted Pyrrolidines .
Rajender Reddy Leleti* et. al.
J. Org. Chem. 2010, 75, 2236

Asymmetric synthesis of 2-substituted pyrrolidines by addition of Grignard reagents to
g-chlorinated N-tert-butanesulfinyl imine.
Rajender Reddy Leleti* et. al.
Chem. Coumn. 2010, 46, 222

An Unexpected Reaction of Arenesulfonyl Cyanide with Allylic Alcohols: Preparation of
Trisubstituted Allyl Sulfones.
Rajender Reddy Leleti* et. al.
Angew. Chemie Int. Ed. 2009, 48, 172

Asymmetric Synthesis of Homoallylic Amines Bearing Adjacent Stereogenic Centers by Addition of  Substituted Allylic Zinc Reagents to N-tert-Butanesulfinyl Imines.
Rajender Reddy Leleti* et. al.
Organic Lett.  2008, 10, 3109

Novel Acetoxylation and C-C Coupling Reactions at Unactivated Positions in-Amino Acid      Derivatives.
L. Rajender Reddy,  E. J. Corey et. al.
Organic Lett. 2006, 8(15), 3391-3394

An Efficient Method for Selective Introduction of Substituents as C(5) of Isoleucine and other a-Amino Acids
L. Rajender Reddy,  E. J. Corey et. al.
Organic Lett  2006, 8(13), 2819-2821

A Novel Bicyclization  Reaction Leading to a fused b-Lactone
L. Rajender Reddy, E. J. Corey et. al.
Organic Lett. 2006, 8(8), 1717-1719

An Efficient, Stereaocontrolled Synthesis of a Potent Omuralide-Salinosporin Hybrid for Selective Proteasome Inhibition.
L. Rajender Reddy, E. J. Corey et. al.
J. Am. Chem. Soc. 2005, 127(25), 8974-8976

A New Synthetic Route for the Enantioselective Total Synthesis of Salinosporamide A and Biologically Active Analogs.
L. Rajender Reddy, E. J. Corey et.al.
Organic Lett. 2005, 7(13), 2699-2701

Simple Enantiospecific Syntheses of the C(2)-Diastereomers of Omuralide and 3-Methylomuralide.
L. Rajender Reddy, E. J. Corey et. al.
Organic Lett. 2005, 7(13), 2703-2705        

A Simple Stereocontrolled Synthesis of Salinosporamide A.
L. Rajender Reddy, E. J. Corey et. al
J. Am. Chem. Soc. 2004, 126 (20), 6230-6231

Functionalized Chiral Vinyl Aminosulfoxonium Salts: Asymmetric Synthesis and  Application to   the Synthesis of Enantiopure Unsaturated Prolines,b,g-Dehydro Amino Acids, and Cyclopentanoid Keto Aminosulfoxonium Ylides
H. -J. Gais, Leleti Rajender Reddy et. al.
J. Am. Chem. Soc. 2006, 128(22), 7360-7373

Asymmetric Synthesis of 2,3-Dihydrofurans and of Unsaturated Tetrahydrofurans Through a-Elimination and Migratory Cyclization of Silyloxy Alkenyl Aminosulfoxonium Salts. Generation and Intramolecular O, Si-Bond Insertion of Chiral Disubstituted b-Silyloxy Alkylidene Carbenes.
H. -J. Gais, L. Rajender Reddy et. al.
J. Am. Chem. Soc. 2004, 126(15), 4859-4864

Asymmetric Synthesis of anti Homopropargylic Alcohols From Aldehydes and Chiral Sulfuonimidoyl Substituted Bis(allyl)titanium Complexes Through  Generation and Elimination of Novel Alkylidenecarbene  (Dimethylamino)sulfoxonium Ylides.
L. Rajender Reddy,  H. -J. Gais, et.al.
J. Am. Chem. Soc. 2002, 124(35), 10427-10434

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PATENTS